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Adamu Uzairu Selected Research

Neoplasms (Cancer)

10/2023Virtual screening, pharmacokinetic, and DFT studies of anticancer compounds as potential V600E-BRAF kinase inhibitors.
10/2023New flavone-based arylamides as potential V600E-BRAF inhibitors: Molecular docking, DFT, and pharmacokinetic properties.
2/2023In silico analysis of noscapine compounds as anti-tumor agents targeting the tubulin receptor.
1/2023Modelling PIP4K2A inhibitory activity of 1,7-naphthyridine analogues using machine learning and molecular docking studies.
1/2022Theoretical modeling and design of some pyrazolopyrimidine derivatives as Wolbachia inhibitors, targeting lymphatic filariasis and onchocerciasis.
4/2020Computational studies of a series of 2-substituted phenyl-2-oxo-, 2-hydroxyl- and 2-acylloxyethylsulfonamides as potent anti-fungal agents.
3/2020QSAR modelling and molecular docking studies for anti-cancer compounds against melanoma cell line SK-MEL-2.

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Adamu Uzairu Research Topics

Disease

7Neoplasms (Cancer)
10/2023 - 03/2020
5Human Influenza (Influenza)
08/2023 - 01/2022
3Melanoma (Melanoma, Malignant)
10/2023 - 03/2020
2Schistosomiasis (Bilharziasis)
04/2024 - 01/2024
2Leishmaniasis
11/2023 - 01/2023
2Breast Neoplasms (Breast Cancer)
08/2023 - 12/2020
2Mental Disorders (Mental Disorder)
07/2020 - 10/2019
1Malaria
04/2024
1Type 2 Diabetes Mellitus (MODY)
01/2024
1Visceral Leishmaniasis (Kala Azar)
11/2023
1Pancreatic Neoplasms (Pancreatic Cancer)
02/2023
1Rheumatoid Arthritis
01/2023
1Autoimmune Diseases (Autoimmune Disease)
01/2023
1Chronic Disease (Chronic Diseases)
01/2023
1Type 1 Diabetes Mellitus (Autoimmune Diabetes)
01/2023
1COVID-19
12/2022
1Schizophrenia (Dementia Praecox)
07/2020
1Non-Small-Cell Lung Carcinoma (Carcinoma, Non-Small Cell Lung)
02/2020
1Prostatic Neoplasms (Prostate Cancer)
01/2020
1Psychotic Disorders (Schizoaffective Disorder)
10/2019
1Tuberculosis (Tuberculoses)
01/2018
1Epilepsy (Aura)
01/2017

Drug/Important Bio-Agent (IBA)

4Neuraminidase (Sialidase)IBA
08/2023 - 01/2022
3VaccinesIBA
04/2024 - 01/2023
3LigandsIBA
04/2024 - 07/2020
3EnzymesIBA
01/2024 - 12/2022
2Praziquantel (Biltricide)FDA Link
04/2024 - 01/2024
2Proteins (Proteins, Gene)FDA Link
01/2023 - 03/2020
1Peptide Elongation Factor 2 (EF-2)IBA
04/2024
17-keto-sempervirolIBA
01/2024
1OxamniquineFDA Link
01/2024
1AmylasesFDA Link
01/2024
1Organoselenium CompoundsIBA
11/2023
1Protein Kinases (Protein Kinase)IBA
10/2023
1Phosphotransferases (Kinase)IBA
10/2023
1Hemagglutinins (Hemagglutinin)IBA
05/2023
1Noscapine (Narcotine)IBA
02/2023
1TubulinIBA
02/2023
1Reactive Oxygen Species (Oxygen Radicals)IBA
01/2023
1Protein Tyrosine PhosphatasesIBA
01/2023
1SARS-CoV-2 3C-like proteinaseIBA
01/2023
1cyclohexanoneIBA
01/2023
1Protein Isoforms (Isoforms)IBA
01/2023
1DNA-Directed RNA Polymerases (RNA Polymerase)IBA
12/2022
1Peptide Hydrolases (Proteases)FDA Link
12/2022
1Transcription Factors (Transcription Factor)IBA
12/2022
1Deubiquitinating EnzymesIBA
01/2022
1Doxycycline (Periostat)FDA LinkGeneric
01/2022
1Estrogens (Estrogen)FDA Link
12/2020
1Antipsychotic Agents (Antipsychotics)IBA
07/2020
1Dopamine Plasma Membrane Transport Proteins (Dopamine Transporter)IBA
07/2020
1SulfonamidesIBA
04/2020
1QuinazolinesIBA
02/2020
1PiperazineIBA
01/2020
1Norepinephrine Plasma Membrane Transport Proteins (Norepinephrine Transporter)IBA
10/2019
1Norepinephrine (Noradrenaline)FDA LinkGeneric
10/2019
1Neurotransmitter Agents (Neurotransmitter)IBA
10/2019
1CytochromesIBA
01/2018
1cytochrome P-450 CYP121IBA
01/2018
1VigabatrinFDA Link
01/2017

Therapy/Procedure

4Therapeutics
11/2023 - 01/2022